Molecule Details
InChIKeyHAZIGHWLODGDFY-UHFFFAOYSA-N
Compound NameN-[3-chloro-4-(9-oxo-8,11-dihydro-7H-pyrrolo[2,1-c][1,4]benzodiazepine-5-carbonyl)phenyl]-5-fluoro-2-methylbenzamide
Canonical SMILESCc1ccc(F)cc1C(=O)Nc1ccc(C(=O)N2C=C3CCC(=O)N3Cc3ccccc32)c(Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30518 AVPR2 Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P30559 OXTR Homo sapiens Human PF00001 6.0 IC50 ChEMBL;BindingDB
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 6.0 IC50 ChEMBL;BindingDB