Target not found.
Molecule Details
InChIKeyHATRKFPXWDUKPL-UHFFFAOYSA-N
Compound Name2-[4-[3-Methoxy-4-[[7-[2-[methyl(methylsulfonyl)amino]phenyl]pyrrolo[2,1-f][1,2,4]triazin-2-yl]amino]phenyl]piperidin-1-yl]acetamide
Canonical SMILESCOc1cc(C2CCN(CC(N)=O)CC2)ccc1Nc1ncc2ccc(-c3ccccc3N(C)S(C)(=O)=O)n2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UM73 ALK Homo sapiens Human PF12810 PF00629 PF07714 7.5 IC50 ChEMBL;BindingDB
P06748 NPM1 Homo sapiens Human PF16276 PF03066 7.1 IC50 ChEMBL
P06213 INSR Homo sapiens Human PF00757 PF17870 PF07714 PF01030 6.3 IC50 ChEMBL;BindingDB