Molecule Details
InChIKeyHAKDXLDJTCFTIE-UHFFFAOYSA-N
Compound NameN-hydroxy-N-[1-(4-hydroxyiminocyclohexyl)-2-[4-[(2-methylquinolin-4-yl)methoxy]phenyl]sulfonylethyl]formamide
Canonical SMILESCc1cc(COc2ccc(S(=O)(=O)CC(C3CCC(=NO)CC3)N(O)C=O)cc2)c2ccccc2n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.18
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P78536 ADAM17 Homo sapiens Human PF16698 PF00200 PF13574 8.1 IC50 ChEMBL
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 6.3 IC50 ChEMBL
P18843 nadE Escherichia coli (strain K12) Pathogen PF02540 Clinical TTD_MultiTarget TTD_MultiTarget