Molecule Details
InChIKeyHAHWOBDKTAQBFE-INIZCTEOSA-N
Compound Name(S)-2-{4-[2-(2-Amino-4-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-ethyl]-benzoylamino}-pentanedioic acid
Canonical SMILESCCc1nc(N)nc2[nH]cc(CCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.04
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.0 IC50 ChEMBL;BindingDB
B0BL08 dfrA17 Escherichia coli Pathogen PF00186 6.0 IC50 BindingDB
P0ABQ4 folA Escherichia coli (strain K12) Pathogen PF00186 6.0 IC50 ChEMBL