Molecule Details
InChIKeyHACFIQPIDCCMMT-FQEVSTJZSA-N
Compound Name4-[4-[2-[(2S)-1-isoquinolin-4-ylsulfonylpyrrolidin-2-yl]ethyl]piperazin-1-yl]-3H-1,3-benzoxazol-2-one
Canonical SMILESO=c1[nH]c2c(N3CCN(CC[C@@H]4CCCN4S(=O)(=O)c4cncc5ccccc45)CC3)cccc2o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P34969 HTR7 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB