Molecule Details
InChIKeyGZRYYCJNHOUUOX-VIFPVBQESA-N
Compound Name4-[4-[(3S)-pyrrolidin-3-yl]sulfonyl-3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl]-1H-benzimidazole-2-carboxylic acid
Canonical SMILESNS(=O)(=O)c1c(S(=O)(=O)[C@H]2CCNC2)ccc(-c2cccc3nc(C(=O)O)[nH]c23)c1-c1nn[nH]n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.05
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.3 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.3 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.5 IC50 BindingDB