Molecule Details
InChIKeyGZQAVBWKRJZVED-DIMJTDRSSA-N
Compound NameN-[(3S)-1-carbamimidoyl-2-hydroxypiperidin-3-yl]-2-[3-(methylsulfamoylamino)-2-oxo-4-(2-phenylethyl)-1-pyridinyl]acetamide
Canonical SMILESCNS(=O)(=O)Nc1c(CCc2ccccc2)ccn(CC(=O)N[C@H]2CCCN(C(=N)N)C2O)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 7.3 IC50 ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 7.0 IC50 ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 6.6 IC50 ChEMBL;BindingDB