Molecule Details
InChIKeyGYQFUHZEIRPWAL-INIZCTEOSA-N
Compound NameN-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[6-[(3S)-3-fluoropyrrolidin-1-yl]-3-pyridinyl]acetamide
Canonical SMILESO=C(Cc1ccc(N2CC[C@H](F)C2)nc1)Nc1ccn(Cc2ccc(F)c(F)c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43497 CACNA1G Homo sapiens Human PF00520 8.6 IC50 ChEMBL;BindingDB
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.3 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 7.7 IC50 ChEMBL;BindingDB