Molecule Details
InChIKeyGYFGNZUSQUDKII-HUYHNIRLSA-N
Compound NameAc-c[Cys-Glu-His-D-Nal(2'')-Arg-Trp-Cys]-Pro-Pro-Lys-Asp-NH2
Canonical SMILESCC(=O)C1C(=O)N[C@H](CCC(=O)O)C(=O)N[C@@H](Cc2c[nH]cn2)C(=O)N[C@@H](Cc2ccc3ccccc3c2)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)NC(C(=O)N2CCC[C@H]2C(=O)CN2CCC[C@H]2C(=O)CN[C@@H](CCCCN)C(=O)CN[C@@H](CC(=O)O)C(N)=O)CSSC1(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41968 MC3R Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB