Molecule Details
InChIKeyGYCXQPDCHIDSOF-UHFFFAOYSA-N
Compound Name2-amino-4-chloro-7-[(2,6-difluoro-3-methoxyphenyl)methyl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
Canonical SMILESCOc1ccc(F)c(CN2C(=O)Cc3c(Cl)nc(N)nc32)c1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12931 TRAP1 Homo sapiens Human PF13589 PF00183 6.6 IC50 ChEMBL;BindingDB
P14625 HSP90B1 Homo sapiens Human PF13589 PF00183 6.2 IC50 ChEMBL;BindingDB
P07900 HSP90AA1 Homo sapiens Human PF13589 PF00183 6.0 IC50 ChEMBL;BindingDB