Molecule Details
InChIKeyGYBZVTMKISJGBF-UHFFFAOYSA-N
Compound NameN-(3-(trifluoromethyl)-5-((4-methylpiperazin-1-yl)methyl)phenyl)-3-(2-(pyrazolo[1,5-a]pyrimidin-6-yl)ethynyl)benzamide
Canonical SMILESCN1CCN(Cc2cc(NC(=O)c3cccc(C#Cc4cnc5ccnn5c4)c3)cc(C(F)(F)F)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q08345 DDR1 Homo sapiens Human PF21114 PF00754 PF07714 8.2 IC50 ChEMBL;BindingDB
Q16832 DDR2 Homo sapiens Human PF21114 PF00754 PF07714 7.0 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 6.6 IC50 ChEMBL;BindingDB