Molecule Details
InChIKeyGXSDXKGIICWKIF-FPOVZHCZSA-N
Compound Name1-(2-aminophenyl)-4-[(11S,16R)-6-thia-10,14-diazatetracyclo[8.6.1.05,17.011,16]heptadeca-1(17),2,4-trien-14-yl]butan-1-one
Canonical SMILESNc1ccccc1C(=O)CCCN1CC[C@H]2[C@@H](C1)c1cccc3c1N2CCCS3
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB