Molecule Details
InChIKeyGXMYCNTVOUYSEA-VWLOTQADSA-N
Compound Name4-[4-[8-[(8aS)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2,3-dihydropyrrolo[3,2-g]isoquinoline-1-carbonyl]-5-ethylpyrazol-1-yl]benzonitrile
Canonical SMILESCCc1c(C(=O)N2CCc3cc4ccnc(N5CCN6CCC[C@H]6C5)c4cc32)cnn1-c1ccc(C#N)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB