Molecule Details
InChIKeyGWIPZYBIMCNGCR-MRXNPFEDSA-N
Compound Name4-{[(3R)-1-(6,7-dimethoxyquinazolin-4-yl)pyrrolidin-3-yl]oxy}benzonitrile
Canonical SMILESCOc1cc2ncnc(N3CC[C@@H](Oc4ccc(C#N)cc4)C3)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 7.2 Ki ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 6.7 Ki ChEMBL;BindingDB
Q13370 PDE3B Homo sapiens Human PF00233 6.3 Ki ChEMBL;BindingDB