Molecule Details
InChIKeyGWHLYYZPDPZRIU-UHFFFAOYSA-N
Compound Name2-[2-[4-(azetidin-3-ylsulfonyl)-3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl]phenyl]guanidine
Canonical SMILESN=C(N)Nc1ccccc1-c1ccc(S(=O)(=O)C2CNC2)c(S(N)(=O)=O)c1-c1nn[nH]n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.94
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.3 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 8.2 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 7.4 IC50 BindingDB