Molecule Details
InChIKeyGVYUEZFLXAHJAB-UHFFFAOYSA-N
Compound Name2-[4-(4''-Fluoro-biphenyl-3-ylmethyl)-piperazin-1-yl]-pyrimidine
Canonical SMILESFc1ccc(-c2cccc(CN3CCN(c4ncccn4)CC3)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.3 IC50 ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB