Molecule Details
InChIKeyGVOOLHNJOQWXKE-UHFFFAOYSA-N
Compound Name6-(5-methyl-1H-1,2,3-triazol-1-yl)-3-[5-(piperidin-1-ylmethyl)-1H-indol-2-yl]-1H-indazole
Canonical SMILESCc1cnnn1-c1ccc2c(-c3cc4cc(CN5CCCCC5)ccc4[nH]3)n[nH]c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.76
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14757 CHEK1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P50613 CDK7 Homo sapiens Human PF00069 6.4 IC50 ChEMBL
P51946 CCNH Homo sapiens Human PF16899 PF00134 6.4 IC50 BindingDB