Molecule Details
InChIKeyGVDYJBFFYVHNPA-UHFFFAOYSA-N
Compound Name1-isopropyl-3-(6-(2-methyl-5-(trifluoromethyl)benzyloxy)naphthalen-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
Canonical SMILESCc1ccc(C(F)(F)F)cc1COc1ccc2cc(-c3nn(C(C)C)c4ncnc(N)c34)ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.09
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 6.7 IC50 ChEMBL;BindingDB
Q8MMZ7 PKG Toxoplasma gondii Pathogen PF00027 PF00069 7.3 IC50 BindingDB
Q9BJF5 CDPK1 Toxoplasma gondii Pathogen PF13499 PF00069 7.3 IC50 ChEMBL;BindingDB