Molecule Details
InChIKeyGVBUCTDNZRCASG-JXFKEZNVSA-N
Compound Name(10R,15S)-12-[3-(3,4-difluorophenoxy)propyl]-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-trien-3-one
Canonical SMILESO=C1CN2c3c(cccc3[C@@H]3CN(CCCOc4ccc(F)c(F)c4)CC[C@@H]32)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.36
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 8.7 Ki ChEMBL
P28223 HTR2A Homo sapiens Human PF00001 7.8 Ki ChEMBL
P21728 DRD1 Homo sapiens Human PF00001 6.6 Ki ChEMBL
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 6.3 Ki ChEMBL