Molecule Details
InChIKeyGVBJTHQLULFNPT-QOHCPDRESA-N
Compound Name(1R,5R,13R,17S)-17-{[(2E)-3-(4-chlorophenyl)prop-2-en-1-yl]amino}-4-(cyclopropylmethyl)-10-methoxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-14-one
Canonical SMILESCOc1ccc2c3c1O[C@H]1C(=O)CC[C@@]4(NC/C=C/c5ccc(Cl)cc5)[C@@H](C2)N(CC2CC2)CC[C@]314
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB