Molecule Details
InChIKeyGUWQZSKMUJFZMM-UHFFFAOYSA-N
Compound Name2-{[2-(Trifluoromethoxy)benzoyl]amino}-N-[6-(Trifluoromethyl)-1h-Benzimidazol-2-Yl]-1,3-Thiazole-4-Carboxamide
Canonical SMILESO=C(Nc1nc2ccc(C(F)(F)F)cc2[nH]1)c1csc(NC(=O)c2ccccc2OC(F)(F)F)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P48730 CSNK1D Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P49674 CSNK1E Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB