Molecule Details
InChIKeyGUPLVXQEYAKBCK-UHFFFAOYSA-N
Compound NameN-[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-amine
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ncc5c(n4)CCNC5)ncc3F)cc2n1C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB