Molecule Details
InChIKeyGUOPFGOTTDDCFQ-UHFFFAOYSA-N
Compound Name5-methyl-N-[5-[(2-methyl-3-pyridinyl)oxy]pyrazin-2-yl]-6-(trifluoromethyl)-2,3-dihydroindole-1-carboxamide
Canonical SMILESCc1cc2c(cc1C(F)(F)F)N(C(=O)Nc1cnc(Oc3cccnc3C)cn1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB