Molecule Details
InChIKeyGUJILKGAXBCELS-UHFFFAOYSA-N
Compound Name4-Chloro-2-{4-[2-(7,9-dioxo-8-aza-spiro[4.5]dec-8-yl)-ethyl]-piperazin-1-yl}-benzonitrile
Canonical SMILESN#Cc1ccc(Cl)cc1N1CCN(CCN2C(=O)CC3(CCCC3)CC2=O)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35368 ADRA1B Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB