Molecule Details
InChIKeyGUIGWNGIQKNZBN-HHHXNRCGSA-N
Compound Name(5S)-1-(cyclohexylmethyl)-5-(3,4-dichlorophenyl)-5-[2-(3-morpholin-4-ylazetidin-1-yl)ethyl]piperidin-2-one
Canonical SMILESO=C1CC[C@](CCN2CC(N3CCOCC3)C2)(c2ccc(Cl)c(Cl)c2)CN1CC1CCCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P21452 TACR2 Homo sapiens Human PF00001 9.1 IC50 ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 9.0 Kd ChEMBL