Molecule Details
InChIKeyGUERACYCGKAFOU-NSHDSACASA-N
Compound NameN~4~-(5-Cyclopropyl-1h-Pyrazol-3-Yl)-N~2~-[(1s)-1-(1h-Pyrrolo[3,2-B]pyridin-5-Yl)ethyl]pyrimidine-2,4-Diamine
Canonical SMILESC[C@H](Nc1nccc(Nc2cc(C3CC3)[nH]n2)n1)c1ccc2[nH]ccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13153 PAK1 Homo sapiens Human PF00786 PF00069 7.5 Ki ChEMBL;BindingDB
O75914 PAK3 Homo sapiens Human PF00786 PF00069 7.3 IC50 ChEMBL
Q13177 PAK2 Homo sapiens Human PF00786 PF00069 7.3 IC50 ChEMBL