Molecule Details
InChIKeyGUDPVWCEUPKJOV-UHFFFAOYSA-N
Compound Name4-(2-Methylpropyl)-2-[[4-(trifluoromethoxy)phenyl]methyl]-1,4-dihydroimidazo[5,1-d][1,2,5]thiadiazine 3,3-dioxide
Canonical SMILESCC(C)CC1n2cncc2CN(Cc2ccc(OC(F)(F)F)cc2)S1(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P19099 CYP11B2 Homo sapiens Human PF00067 7.0 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.3 IC50 ChEMBL;BindingDB
P15538 CYP11B1 Homo sapiens Human PF00067 6.3 IC50 ChEMBL;BindingDB