Molecule Details
InChIKeyGTZWWDDACCTQQM-UHFFFAOYSA-N
Compound Name3-{5-[(tert-butylamino)methyl]-1H-pyrazol-3-yl}-1-{5-oxo-1H,2H,3H,5H,9bH-benzo[a]pyrrolizin-9-yl}urea
Canonical SMILESCC(C)(C)NCc1cc(NC(=O)Nc2cccc3c2C2CCCN2C3=O)[nH]n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.2 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.2 pIC50 TTD_MultiTarget