Molecule Details
InChIKeyGTTSANJRVQIGFM-UHFFFAOYSA-N
Compound Name4-[[1-[3-[(3,4-Difluorobenzoyl)amino]phenyl]-3-methoxypropyl]amino]quinazoline-8-carboxamide
Canonical SMILESCOCCC(Nc1ncnc2c(C(N)=O)cccc12)c1cccc(NC(=O)c2ccc(F)c(F)c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.7 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.7 IC50 ChEMBL;BindingDB