Molecule Details
InChIKeyGTLGKZJPNAWIBT-UHFFFAOYSA-N
Compound Nameethyl (6-(6-(4-chlorophenyl)-3-cyclopropyl-1-methyl-4-oxopyrrolo[3,4-c]pyrazol-5-(1H,4H,6H)-yl)-3-methyl-[1,2,4]triazolo[4,3-a]pyridin-8-yl)carbamate
Canonical SMILESCCOC(=O)Nc1cc(N2C(=O)c3c(C4CC4)nn(C)c3C2c2ccc(Cl)cc2)cn2c(C)nnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.7 IC50 ChEMBL;BindingDB
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.6 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.6 IC50 ChEMBL;BindingDB