Molecule Details
InChIKeyGTGNAUXPRWWJOU-FQEVSTJZSA-N
Compound Name(S)-benzyl 1-(2-(4-methoxyphenyl)thiazol-4-yl)-5-(sulfamoylamino)pentylcarbamate
Canonical SMILESCOc1ccc(-c2nc([C@H](CCCCNS(N)(=O)=O)NC(=O)OCc3ccccc3)cs2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.31
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.3 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.3 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.3 pIC50 TTD_MultiTarget