Molecule Details
InChIKeyGTAKUJFUJVMIPM-LBPRGKRZSA-N
Compound Name4-N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-N-methyl-2-N-[(1S)-1-(1H-pyrrolo[3,2-b]pyridin-5-yl)ethyl]pyrimidine-2,4-diamine
Canonical SMILESC[C@@H](c1ccc2[nH]ccc2n1)N(C)c1nccc(Nc2cc(C3CC3)[nH]n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.99
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13153 PAK1 Homo sapiens Human PF00786 PF00069 7.7 Ki ChEMBL;BindingDB
O75914 PAK3 Homo sapiens Human PF00786 PF00069 6.6 IC50 ChEMBL
Q13177 PAK2 Homo sapiens Human PF00786 PF00069 6.6 IC50 ChEMBL