Molecule Details
InChIKeyGSWYQMZWPSIFDH-UHFFFAOYSA-N
Compound Name4-[[3-(Dimethylamino)-1-[5-[(2-fluoro-4-methoxybenzoyl)amino]cyclohexa-1,5-dien-1-yl]propyl]amino]quinazoline-8-carboxamide
Canonical SMILESCOc1ccc(C(=O)NC2=CC(C(CCN(C)C)Nc3ncnc4c(C(N)=O)cccc34)=CCC2)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.7 IC50 ChEMBL;BindingDB