Molecule Details
InChIKeyGSQMITXEUGIGFD-UHFFFAOYSA-N
Compound Name3-Methyl-5-oxido-8-(pyridin-4-ylmethoxy)pyrazolo[5,1-c][1,2,4]benzotriazin-5-ium
Canonical SMILESCc1cnn2c1n[n+]([O-])c1ccc(OCc3ccncc3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14867 GABRA1 Homo sapiens Human PF02931 PF02932 7.6 Ki ChEMBL;BindingDB
P18507 GABRG2 Homo sapiens Human PF02931 PF02932 7.6 Ki ChEMBL
P47870 GABRB2 Homo sapiens Human PF02931 PF02932 7.6 Ki ChEMBL