Molecule Details
InChIKeyGSPMAICRXXSRDC-QAQDUYKDSA-N
Canonical SMILESCCO[C@H]1C[C@H](NC(=O)c2ccc(OCc3c(-c4ccc(C)nc4)noc3C)nn2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.06
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14867 GABRA1 Homo sapiens Human PF02931 PF02932 8.1 Ki ChEMBL;BindingDB
P31644 GABRA5 Homo sapiens Human PF02931 PF02932 8.1 Ki BindingDB