Molecule Details
InChIKeyGRTPVLUWVUWRRC-UHFFFAOYSA-N
Compound Name9-dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one
Canonical SMILESCCc1ccc(-n2c(C)nc3c(sc4nccc(N(C)C)c43)c2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13255 GRM1 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 7.4 IC50 ChEMBL;BindingDB
P41594 GRM5 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 6.5 IC50 ChEMBL;BindingDB