Molecule Details
InChIKeyGRKGCIUUSLKRTB-UHFFFAOYSA-N
Compound Name6-(((1-(4-cyanobenzyl)-1H-imidazol-5-yl)methoxy)methyl)-4''-ethoxybiphenyl-3-carbonitrile
Canonical SMILESCCOc1ccc(-c2cc(C#N)ccc2COCc2cncn2Cc2ccc(C#N)cc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.92
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.9 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.9 IC50 ChEMBL;BindingDB