Molecule Details
InChIKeyGRBADRHZGYZJTH-UHFFFAOYSA-N
Compound Name4-[1-[3-[(2-Methoxypyridine-4-carbonyl)amino]cyclohexa-1,3-dien-1-yl]ethylamino]quinazoline-8-carboxamide
Canonical SMILESCOc1cc(C(=O)NC2=CCCC(C(C)Nc3ncnc4c(C(N)=O)cccc34)=C2)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.3 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.5 IC50 ChEMBL;BindingDB