Molecule Details
InChIKeyGQCLNKPNLVDVKR-SJLPKXTDSA-N
Compound Name2-[(3R,6R)-6-methyl-1-[2-methyl-6-(triazol-2-yl)benzoyl]piperidin-3-yl]oxypyridine-4-carbonitrile
Canonical SMILESCc1cccc(-n2nccn2)c1C(=O)N1C[C@H](Oc2cc(C#N)ccn2)CC[C@H]1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O43614 HCRTR2 Homo sapiens Human PF00001 PF03827 8.6 Ki ChEMBL;BindingDB
O43613 HCRTR1 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB