Molecule Details
InChIKeyGPSNGZQIELJYAX-UHFFFAOYSA-N
Compound Name6-[2-[4-(2-methylquinolin-5-yl)oxypiperidin-1-yl]ethyl]-4H-1,4-benzoxazin-3-one
Canonical SMILESCc1ccc2c(OC3CCN(CCc4ccc5c(c4)NC(=O)CO5)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB