Molecule Details
InChIKeyGPRHHSZIXIDKDN-OAHLLOKOSA-N
Compound Name4-Amino-N-{(2R)-3-[4-(3,4-dichlorophenoxy)piperidin-1-yl]-2-hydroxypropyl}-3-methoxybenzamide
Canonical SMILESCOc1cc(C(=O)NC[C@@H](O)CN2CCC(Oc3ccc(Cl)c(Cl)c3)CC2)ccc1N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P51677 CCR3 Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P35367 HRH1 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.6 IC50 ChEMBL;BindingDB