Molecule Details
InChIKeyGPJBNWXFJJEFAT-RDGDOILBSA-N
Compound Name17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4''-methyl)benzamido]morphinan-oxalate
Canonical SMILESCc1ccc(C(=O)N[C@@H]2CC[C@@]3(O)[C@H]4Cc5ccc(O)c6c5[C@@]3(CCN4CC3CC3)[C@H]2O6)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 10.4 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 9.5 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB