Molecule Details
InChIKeyGPDVHOTUPZYYBA-UHFFFAOYSA-N
Compound NameMaleimide derivative, 13
Canonical SMILESO=C1NC(=O)C(c2c[nH]c3ccccc23)=C1c1nc(N2CCOCC2)nc2ccccc12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.1
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.1 pIC50 TTD_MultiTarget
Q05655 PRKCD Homo sapiens Human PF00130 PF21494 PF00069 PF00433 6.1 IC50 ChEMBL;BindingDB