Molecule Details
InChIKeyGOURHBOOQWGQNN-UHFFFAOYSA-N
Compound Name1-[6-(3-methyl-2H-pyrazolo[3,4-c]pyridin-5-yl)pyrazin-2-yl]piperidin-4-amine
Canonical SMILESCc1n[nH]c2cnc(-c3cncc(N4CCC(N)CC4)n3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.2 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.8 Ki ChEMBL;BindingDB