Molecule Details
InChIKeyGOOYSJIWTIHOGW-UHFFFAOYSA-N
Compound Name4-[3-(2-Methoxy-pyridin-3-yl)-pyrazolo[1,5-a]pyrimidin-5-yl]-piperazine-1-carboxylic acid isopropyl ester
Canonical SMILESCOc1ncccc1-c1cnn2ccc(N3CCN(C(=O)OC(C)C)CC3)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.37
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q2M2I8 AAK1 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
Q9NSY1 BMP2K Homo sapiens Human PF15282 PF00069 7.5 IC50 BindingDB
O14976 GAK Homo sapiens Human PF00069 PF10409 6.1 IC50 BindingDB