Molecule Details
InChIKeyGNAXCGUONRASLS-UHFFFAOYSA-N
Compound Name6-[1-(6-piperazin-1-yl-2-pyridinyl)pyrazolo[4,3-c]pyridin-6-yl]-1H-pyrazin-2-one
Canonical SMILESO=c1cncc(-c2cc3c(cn2)cnn3-c2cccc(N3CCNCC3)n2)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.2 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.8 Ki ChEMBL;BindingDB