Molecule Details
InChIKeyGNAOSQHBSOBWJQ-UHFFFAOYSA-N
Compound Name2-[4-(4-Chlorophenyl)phenyl]sulfonyl-4-(1,3-dioxoisoindol-2-yl)butanoic acid
Canonical SMILESO=C(O)C(CCN1C(=O)c2ccccc2C1=O)S(=O)(=O)c1ccc(-c2ccc(Cl)cc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.29
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.7 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 7.8 IC50 ChEMBL;BindingDB