Molecule Details
InChIKeyGMOGCDFLNRXOJV-UHFFFAOYSA-N
Compound NameN-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)-7-(1H-pyrazol-4-yl)quinazolin-2-amine
Canonical SMILESc1cc(-n2cnc(N3CCOCC3)n2)ccc1Nc1ncc2ccc(-c3cn[nH]c3)cc2n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.21
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P05412 JUN Homo sapiens Human PF00170 PF03957 6.9 IC50 ChEMBL;BindingDB