Molecule Details
InChIKeyGMKWDFMANHJRNB-UHFFFAOYSA-N
Compound Name5-hydroxy-8-[4-[4-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]butyl]-1,4-diazepan-1-yl]-4H-1,4-benzoxazin-3-one
Canonical SMILESO=C1CCc2ccc(OCCCCN3CCCN(c4ccc(O)c5c4OCC(=O)N5)CC3)cc2N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB