Molecule Details
InChIKeyGMIKNOQZLHKCFH-UHFFFAOYSA-N
Compound Name2-{2-[(3,4-Difluorophenoxy)methyl]-5-Methoxypyridin-4-Yl}-1,5,6,7-Tetrahydro-4h-Pyrrolo[3,2-C]pyridin-4-One
Canonical SMILESCOc1cnc(COc2ccc(F)c(F)c2)cc1-c1cc2c([nH]1)CCNC2=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P48730 CSNK1D Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P78368 CSNK1G2 Homo sapiens Human PF12605 PF00069 6.7 IC50 ChEMBL;BindingDB
P48729 CSNK1A1 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB